SCHEMBL7599430

SCHEMBL7599430

COc1cccc(C(=CC2=NCCN2C(=O)O)c2ccncc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 3/20 0.43
KDM2B Q8NHM5 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1B1 Q16678 1/20 0.42
ABL1 P00519 2/20 0.41
BCR P11274 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MTNR1A P48039 2/20 0.41
MTNR1B P49286 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
GPR6 P46095 1/20 0.41
CYP11B1 P15538 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599426 1.00 NPC1 (0.43) NPC1ALDH1A1KDM2BHPGDKMT2A
SCHEMBL7549453 0.88 KMT2A (0.42) NPC1ALDH1A1KDM2BHPGDKMT2A
SCHEMBL7549457 0.88 KMT2A (0.42) NPC1ALDH1A1KDM2BHPGDKMT2A
SCHEMBL7549956 0.88 KMT2A (0.42) NPC1ALDH1A1KDM2BHPGDKMT2A
SCHEMBL7555175 0.73 NISCH (0.46) NPC1KMT2ACYP1A2CYP2D6CYP1A1
SCHEMBL7555168 0.73 NISCH (0.46) NPC1KMT2ACYP1A2CYP2D6CYP1A1
SCHEMBL7555183 0.73 NISCH (0.46) NPC1KMT2ACYP1A2CYP2D6CYP1A1
SCHEMBL4029309 0.69 CES2 (0.77) NPC1ALDH1A1HPGDKMT2ACYP1A2
SCHEMBL5216406 0.69 KMT2A (0.72) NPC1ALDH1A1KMT2ACYP1A2CYP2D6
SCHEMBL4068210 0.66 KMT2A (0.73) ALDH1A1KDM2BKMT2AL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002038559-A1 1,3-DIAZAHETEROCYCLIC COMPOUNDS AND THEIR USE AS ORAL HYPOGLYCAEMIC AGENTS NOVO NORDISK A/S (DK) 2002-05-16 WO disclosed