SCHEMBL7599591

SCHEMBL7599591

CC(CCC(=O)O)(c1ccc(OCc2ncccn2)cc1)c1ccc(OCc2ncccn2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.57
ESR1 P03372 1/20 0.57
CYP3A4 P08684 1/20 0.57
ESR2 Q92731 1/20 0.57
CHEK1 O14757 1/20 0.44
FYN P06241 1/20 0.44
PDGFRB P09619 1/20 0.44
PIM1 P11309 1/20 0.44
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
GRK5 P34947 1/20 0.44
MAP2K2 P36507 1/20 0.44
MAPK8 P45983 1/20 0.44
CDK8 P49336 1/20 0.44
RPS6KA3 P51812 1/20 0.44
PRKX P51817 1/20 0.44
JAK3 P52333 1/20 0.44
LIMK1 P53667 1/20 0.44
BTK Q06187 1/20 0.44
TYRO3 Q06418 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7594842 0.86 ALDH1A1 (0.54) ALDH1A1ESR1CYP3A4ESR2MAPK14
SCHEMBL7594540 0.85 ALDH1A1 (0.47) ALDH1A1ESR1CYP3A4ESR2CHEK1
SCHEMBL7596217 0.85 ALDH1A1 (0.52) ALDH1A1ESR1CYP3A4ESR2MAPK14
SCHEMBL28205576 0.83 ALDH1A1 (0.60) ALDH1A1ESR1CYP3A4ESR2NR4A2
SCHEMBL6440668 0.79 CYSLTR1 (0.67) FFAR1CYSLTR2CYSLTR1AKR1B1
SCHEMBL30538032 0.79 CYSLTR1 (0.67) FFAR1CYSLTR2CYSLTR1AKR1B1
SCHEMBL7595880 0.79 ALDH1A1 (0.46) ALDH1A1ESR1CYP3A4ESR2MAPK14
SCHEMBL3048632 0.78 CYSLTR1 (0.66) FFAR1CYSLTR2CYSLTR1AKR1B1
SCHEMBL3048640 0.78 CYSLTR1 (0.66) FFAR1CYSLTR2CYSLTR1AKR1B1
SCHEMBL7595258 0.78 CYSLTR1 (0.66) FFAR1CYSLTR2CYSLTR1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0862557-B1 SYMMETRICAL bis-HETEROARYLMETHOXYPHENYLALKYL CARBOXYLATES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LAB (US) 2002-11-27 EP disclosed
US-5843968-A Symmetrical bis-heteroarylmethoxy-phenylalkyl carboxylates as inhibitors of leukotriene biosynthesis ABBOTT LABORATORIES (US) 1998-12-01 US disclosed
US-5795900-A Symmetrical bis-heteroaryl-methoxy-phenylalkyl carboxylates as inhibitors of leukotriene biosynthesis ABBOTT LABORATORIES (US) 1998-08-18 US disclosed