SCHEMBL7602762

SCHEMBL7602762

C=C(O)CCc1cccc(NC(=O)[C@H](c2ccc(Cn3cc(C(F)(F)F)ccc3=O)cc2)[C@@H](C)C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
POLB P06746 1/20 0.49
KMT2A Q03164 1/20 0.46
MAPT P10636 5/20 0.45
LMNA P02545 3/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
HTT P42858 1/20 0.41
S1PR2 O95136 1/20 0.40
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 2/20 0.39
NPC1 O15118 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703077 0.94 CYP1A2 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3698632 0.94 CYP1A2 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3704557 0.89 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3694470 0.89 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7601286 0.84 KCNJ6 (0.39) KMT2A
SCHEMBL7602084 0.77 IDH1 (0.34) KMT2AMAPTLMNA
SCHEMBL1178416 0.77 KMT2A (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7605713 0.77 KMT2A (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1177620 0.77 KMT2A (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1178424 0.77 KMT2A (0.55) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed