SCHEMBL7604313

SCHEMBL7604313

CCC(N)c1c[nH]c2c(OCC(=O)N(CC)CC)cccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
ADRB3 P13945 2/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
GLA P06280 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5480473 0.82 TSHR (0.53) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL5480477 0.82 TSHR (0.53) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL5857882 0.81 TSHR (0.51) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL5859950 0.81 TSHR (0.51) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL7636048 0.79 TSHR (0.45) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL7604319 0.77 TSHR (0.52) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL7593268 0.76 ADRB3 (0.46) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL5479233 0.74 ADRB3 (0.54) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL5485060 0.74 ADRB3 (0.54) TSHRADRB3ADRB2ADRB1BCHE
SCHEMBL5858588 0.72 TSHR (0.48) TSHRADRB3ADRB2ADRB1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6458824-B1 (3-((2R)-(((2R)-(3-CHLOROPHENYL)-2-HYDROXYETHYL)AMINO)PROPYL)-1H-INDOL-7-YLOXY)ACETIC ACID CRYSTAL SOLIDS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2002-10-01 US disclosed
EP-1235801-A2 SOLID PHARMACEUTICAL PREPARATION Dainippon Pharmaceutical Co., Ltd. (JP) 2002-09-04 EP disclosed
WO-2001040182-A2 SOLID PHARMACEUTICAL PREPARATION DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2001-06-07 WO disclosed