SCHEMBL7604442

SCHEMBL7604442

CN(C)CC1=C(c2cccc(O)c2)c2ccc(O)cc2SCC1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 12/20 0.33
HSD17B2 P37059 12/20 0.33
PIK3CA P42336 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
PIM1 P11309 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2B6 P20813 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8016502 0.99 PIK3CA (0.33) HSD17B1HSD17B2PIK3CACHRNB4CHRNA3
SCHEMBL7606364 0.91 ESR1 (0.40) HSD17B1HSD17B2PIK3CACHRNB4CHRNA3
SCHEMBL7610138 0.90 HPGD (0.37) HSD17B1HSD17B2PIK3CACHRNB4CHRNA3
Hydrochloric Acid SCHEMBL8023704 0.90 ESR1 (0.40) HSD17B1HSD17B2PIK3CAESR1ESR2
Hydrochloric Acid SCHEMBL8016754 0.89 HPGD (0.36) HSD17B1HSD17B2PIK3CACHRNB4CHRNA3
SCHEMBL7615755 0.89 KDM4E (0.45) HSD17B1HSD17B2ESR1ESR2CYP3A4
Hydrochloric Acid SCHEMBL8020664 0.88 KDM4E (0.44) HSD17B1HSD17B2ALDH1A1ESR1ESR2
SCHEMBL7588665 0.80 ESR1 (0.40) HSD17B1HSD17B2CHRNB4CHRNA3ESR1
SCHEMBL7609641 0.79 ADRA2A (0.36) HSD17B1HSD17B2PIK3CAALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8017994 0.79 ESR1 (0.39) HSD17B1HSD17B2CHRNB4CHRNA3ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed