SCHEMBL7605652

SCHEMBL7605652

CN(C)CS[C@H]1COc2ccccc2C1=O

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.48
CYP19A1 P11511 14/20 0.48
SIGMAR1 Q99720 2/20 0.40
HTR1A P08908 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10916938 1.00 MAOB (0.48) MAOBCYP19A1SIGMAR1HTR1APKM
Hydrochloric Acid SCHEMBL10916087 0.99 MAOB (0.47) MAOBCYP19A1SIGMAR1HTR1A
Hydrochloric Acid SCHEMBL10917082 0.82 METAP1 (0.43) MAOBCYP19A1
Hydrochloric Acid SCHEMBL10916524 0.81 CYP19A1 (0.51) MAOBCYP19A1PKM
Hydrochloric Acid SCHEMBL10914965 0.79 DAO (0.39) MAOBCYP19A1
Hydrochloric Acid SCHEMBL10915392 0.79 CYP19A1 (0.34) MAOBCYP19A1
SCHEMBL7153929 0.78 CYP19A1 (0.56) MAOBCYP19A1SIGMAR1PKMTSHR
SCHEMBL6775349 0.76 MAOB (0.61) MAOBCYP19A1SIGMAR1HTR1A
SCHEMBL7604495 0.76 MAOB (0.61) MAOBCYP19A1SIGMAR1HTR1A
SCHEMBL31073649 0.76 MAOB (0.61) MAOBCYP19A1SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
US-6013809-A ANALGESICS GRUENENTHAL GMBH (DE) 2000-01-11 US disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed