SCHEMBL7606302

SCHEMBL7606302

Nc1ccc(Sc2ccc(Cl)cc2Cl)c(C(F)(F)F)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 4/20 0.68
ICAM1 P05362 4/20 0.68
ITGAL P20701 4/20 0.68
PDE7A Q13946 3/20 0.47
TSHR P16473 3/20 0.44
GLA P06280 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
RHEB Q15382 2/20 0.41
CYP3A4 P08684 3/20 0.38
KDM4E B2RXH2 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTR1A P08908 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR3A P46098 1/20 0.38
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL709679 0.85 GAA (0.59) ITGB2ICAM1ITGALPDE7ATSHR
SCHEMBL7610324 0.83 ITGB2 (0.96) ITGB2ICAM1ITGALPDE7ATSHR
Hydrochloric Acid SCHEMBL7637698 0.81 ITGB2 (1.00) ITGB2ICAM1ITGALPDE7ATSHR
SCHEMBL28351861 0.81 CYP2D6 (0.43) ITGB2ICAM1ITGALPDE7ATSHR
SCHEMBL7607010 0.79 ITGB2 (0.74) ITGB2ICAM1ITGALPDE7ATSHR
SCHEMBL30761014 0.76 PDE7A (0.63) PDE7ATSHRGLAPOLBGAA
SCHEMBL7610002 0.76 PDE7A (0.59) ITGB2ICAM1ITGALPDE7AHSD17B10
SCHEMBL30574189 0.75 TSHR (0.61) TSHRGLAPOLBGAACYP3A4
SCHEMBL203216 0.75 TSHR (0.61) TSHRGLAPOLBGAACYP3A4
SCHEMBL7187676 0.75 ITGB2 (0.80) ITGB2ICAM1ITGALPDE7ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165504-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2002-01-02 EP disclosed
WO-2000059878-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2000-10-12 WO disclosed