SCHEMBL7607010

SCHEMBL7607010

Nc1ccc(Sc2ccc(Cl)cc2Cl)c(F)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 4/20 0.74
ICAM1 P05362 4/20 0.74
ITGAL P20701 4/20 0.74
PDE7A Q13946 3/20 0.51
KDM4E B2RXH2 2/20 0.43
ATM Q13315 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RHEB Q15382 1/20 0.41
CYP3A4 P08684 4/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
PDE7B Q9NP56 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610324 0.87 ITGB2 (0.96) ITGB2ICAM1ITGALPDE7AKDM4E
Hydrochloric Acid SCHEMBL7637698 0.85 ITGB2 (1.00) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL7605654 0.83 ITGB2 (0.59) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL7187676 0.79 ITGB2 (0.80) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL3165346 0.79 ITGB2 (0.72) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL7606302 0.79 ITGB2 (0.68) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL7610177 0.79 ITGB2 (0.79) ITGB2ICAM1ITGALPDE7AKDM4E
Hydrochloric Acid SCHEMBL7604738 0.78 ITGB2 (0.77) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL7610151 0.76 ITGB2 (0.74) ITGB2ICAM1ITGALPDE7AKDM4E
SCHEMBL2030464 0.75 PDE7A (0.69) ITGB2ICAM1ITGALPDE7AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165504-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2002-01-02 EP disclosed
WO-2000059878-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2000-10-12 WO disclosed