SCHEMBL7607570

SCHEMBL7607570

CCCn1c(=O)n(COCC)c(=O)c2[nH]cnc21

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 18/20 0.79
PDE4B Q07343 18/20 0.79
PDE4C Q08493 18/20 0.79
PDE4D Q08499 18/20 0.79
ADORA2A P29274 12/20 0.79
ADORA2B P29275 10/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455363 0.88 ADORA2A (0.72) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL515771 0.87 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
Ammonia Solution, Strong SCHEMBL10420651 0.86 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL4623455 0.84 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL5400933 0.83 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7603090 0.83 ADORA2A (0.72) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7608673 0.83 PDE4A (0.85) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3842077 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381259 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9765669 0.81 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214992-B1 THEOPHYLLINE DERIVATIVES HAVING AT LEAST ONE ETHER FUNCTION IN METHYL RADICAL; XANTHINE COMPOUNDS WITH THIS SUBSTITUTION PATTERN USED AS ANTISHOCK TREATMENT HOECHST AKTIENGESELLSCHAFT (DE) 2001-04-10 US claimed
EP-0812844-B1 Use of theophyllin derivatives for the treatment and prophylaxis fo shock conditions, novel xanthine compounds and processes for the production thereof HOECHST AG (DE) 2002-10-23 EP disclosed
US-6214992-B1 THEOPHYLLINE DERIVATIVES HAVING AT LEAST ONE ETHER FUNCTION IN METHYL RADICAL; XANTHINE COMPOUNDS WITH THIS SUBSTITUTION PATTERN USED AS ANTISHOCK TREATMENT HOECHST AKTIENGESELLSCHAFT (DE) 2001-04-10 US disclosed
EP-0812844-A2 Use of theophyllin derivatives for the treatment and prophylaxis fo shock conditions, novel xanthine compounds and processes for the production thereof HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-17 EP disclosed