SCHEMBL7608324

SCHEMBL7608324

CCOC(=O)C=Cc1ccc(O)cc1C#N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA14 Q9ULX7 1/20 0.55
MIF P14174 1/20 0.49
TTR P02766 1/20 0.48
DPP4 P27487 1/20 0.48
ESR1 P03372 3/20 0.47
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
CYP3A4 P08684 1/20 0.46
AKR1B10 O60218 6/20 0.45
AKR1B1 P15121 6/20 0.45
MAOB P27338 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14111461 1.00 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL28664848 0.86 TTR (0.45) CA12CA1CA2CA7CA9
SCHEMBL11353377 0.85 TTR (0.44) CA12CA1CA2CA7CA9
SCHEMBL11428624 0.85 MAPT (0.45) CA12CA1CA2CA7CA9
SCHEMBL11428626 0.85 MAPT (0.45) CA12CA1CA2CA7CA9
SCHEMBL11353373 0.85 TTR (0.44) CA12CA1CA2CA7CA9
SCHEMBL4894153 0.84 MIF (0.43) CA12CA1CA2CA7CA9
SCHEMBL4894150 0.84 MIF (0.43) CA12CA1CA2CA7CA9
SCHEMBL16218971 0.83 TTR (0.46) CA12CA1CA2CA7CA9
SCHEMBL2582174 0.82 HSD17B1 (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395919-B1 Calcilytic compounds SMITHKLINE BEECHAM CORPORATION 2002-05-28 US disclosed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP disclosed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed