SCHEMBL7609151

SCHEMBL7609151

N=C(N)CSCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.57
NOS1 P29475 3/20 0.57
NOS3 P29474 1/20 0.57
NOS2 P35228 1/20 0.57
CYP2C19 P33261 1/20 0.47
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NFKB1 P19838 1/20 0.44
CASP3 P42574 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
SLC11A2 P49281 1/20 0.44
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7614580 0.98 IDO1 (0.59) IDO1NOS1NOS3NOS2CYP2C19
SCHEMBL1478837 0.83 MEN1 (0.66) IDO1NOS1NOS3NOS2CYP2C19
Bromide SCHEMBL3375119 0.81 MEN1 (0.63) IDO1NOS1NOS3NOS2CYP2C19
Hydrochloric Acid SCHEMBL5506583 0.81 MEN1 (0.63) IDO1NOS1NOS3NOS2CYP2C19
SCHEMBL7106171 0.81 IDO1 (0.50) IDO1NOS1NOS3NOS2CYP2C19
SCHEMBL499117 0.76 CYP2C19 (0.64) CYP2C19NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL20395222 0.76 CYP2C19 (0.59) CYP2C19NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL206 0.75 CYP2C19 (0.56) IDO1NOS1NOS3NOS2CYP2C19
SCHEMBL721637 0.74 CYP2C19 (0.57) CYP2C19NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL5840786 0.74 CYP2C19 (0.57) CYP2C19NPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724435-B1 AMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2002-08-14 EP claimed
EP-0399856-B1 Pteridin-4 (3H)-ones, processes for their preparation and medicaments containing them LIPHA (FR) 1995-08-09 EP disclosed
US-5270465-A 4(3H)-pteridinone compounds LIPHA, LYONNAISE INDUSTRILLE PHARMACEUTIQUE (FR) 1993-12-14 US disclosed
US-5167949-A Antiallergic LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1992-12-01 US disclosed
EP-0399856-A1 Pteridin-4 (3H)-ones, processes for their preparation and medicaments containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1990-11-28 EP disclosed