SCHEMBL7609158

SCHEMBL7609158

C=CCN(c1ccncc1F)n1ccc2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.66
MAPT P10636 3/20 0.34
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
TGFBR1 P36897 1/20 0.31
TGFBR2 P37173 1/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7621062 0.99 SLC6A2 (0.65) SLC6A2MAPTMKNK1MKNK2TGFBR1
SCHEMBL7610925 0.84 SLC6A2 (0.65) SLC6A2MAPTMKNK1MKNK2TGFBR1
Hydrochloric Acid SCHEMBL7617563 0.83 SLC6A2 (0.64) SLC6A2MAPTMKNK1MKNK2TGFBR1
SCHEMBL8946156 0.82 SLC6A2 (0.49) SLC6A2MAPTMKNK1MKNK2BCHE
SCHEMBL7611649 0.82 SLC6A2 (0.65) SLC6A2BCHE
Hydrochloric Acid SCHEMBL3977692 0.81 SLC6A2 (0.64) SLC6A2BCHE
SCHEMBL9795990 0.80 SLC6A2 (1.00) SLC6A2
SCHEMBL7611577 0.78 SLC6A2 (0.49) SLC6A2BCHE
Hydrochloric Acid SCHEMBL7613979 0.77 SLC6A2 (0.48) SLC6A2BCHE
SCHEMBL9796088 0.76 SLC6A2 (0.44) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840609-B1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS AVENTIS PHARMA INC (US) 2002-06-05 EP claimed
US-5776955-A Use of unsubstituted and substituted n-(pyrrol-1-yl)pyridinamines as anticonvulsant agents HOECHST MARION ROUSSEL, INC. 1998-07-07 US claimed
EP-0840609-A1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-05-13 EP claimed
WO-1997004777-A1 USE OFF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-02-13 WO claimed
EP-0840609-B1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS AVENTIS PHARMA INC (US) 2002-06-05 EP disclosed
US-5776955-A Use of unsubstituted and substituted n-(pyrrol-1-yl)pyridinamines as anticonvulsant agents HOECHST MARION ROUSSEL, INC. 1998-07-07 US disclosed
US-5039811-A Analgesics, antidepressants, memory activators; condensation, reduction HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-13 US disclosed
US-4970218-A ANALGESIC, ANTIDEPRESSANT, MEMORY ENHANCEMENT HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-11-13 US disclosed