SCHEMBL7609174

SCHEMBL7609174

CCC(Sc1cc(Cl)ccc1C#N)c1cccc(NC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 9/20 0.54
CYP2D6 P10635 8/20 0.54
SLC6A2 P23975 8/20 0.54
SLC6A4 P31645 8/20 0.54
KCNH2 Q12809 2/20 0.39
ALDH1A1 P00352 3/20 0.33
LMNA P02545 2/20 0.33
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 3/20 0.32
MAPT P10636 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
VCAM1 P19320 1/20 0.32
CBLB Q13191 2/20 0.31
GAA P10253 2/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
EGFR P00533 1/20 0.31
ERBB2 P04626 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5648745 0.77 SLC6A2 (0.70) NOS2CYP2D6SLC6A2SLC6A4KCNH2
Hydrochloric Acid SCHEMBL5650489 0.76 SLC6A2 (0.68) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL27513304 0.75 NOS2 (0.59) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL6494143 0.74 SLC6A4 (0.72) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL7607981 0.74 NOS2 (0.38) NOS2CYP2D6SLC6A2SLC6A4KCNH2
Hydrochloric Acid SCHEMBL27526759 0.74 NOS2 (0.60) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL6278719 0.74 CYP2D6 (0.41) NOS2CYP2D6SLC6A2SLC6A4ALDH1A1
Hydrochloric Acid SCHEMBL6496956 0.74 SLC6A4 (0.71) NOS2CYP2D6SLC6A2SLC6A4KCNH2
SCHEMBL5653417 0.72 NOS2 (0.81) NOS2CYP2D6SLC6A2SLC6A4KCNH2
Hydrochloric Acid SCHEMBL5652171 0.71 NOS2 (0.79) NOS2CYP2D6SLC6A2SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263718-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP claimed
WO-2001062721-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO claimed
EP-1263718-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062721-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed