SCHEMBL7610074

SCHEMBL7610074

COc1ccc(NC(=O)C=Cc2ccc(C#N)cc2)cc1CCCN(C(C)C)C(C)C

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.54
ACHE P22303 2/20 0.47
CA12 O43570 5/20 0.46
CA9 Q16790 5/20 0.46
MAOB P27338 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
MAOA P21397 1/20 0.46
TRPV1 Q8NER1 3/20 0.46
IMPDH2 P12268 2/20 0.45
IMPDH1 P20839 1/20 0.45
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
BCHE P06276 2/20 0.42
HDAC1 Q13547 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610070 1.00 SLC2A1 (0.54) SLC2A1ACHECA12CA9MAOB
SCHEMBL7610076 0.88 ACHE (0.48) ACHECA12CA9MAOBCA1
SCHEMBL7611221 0.88 SLC2A1 (0.56) SLC2A1ACHECA12CA9CA1
SCHEMBL7615759 0.88 SLC2A1 (0.56) SLC2A1ACHECA12CA9CA1
SCHEMBL7611226 0.88 SLC2A1 (0.56) SLC2A1ACHECA12CA9CA1
SCHEMBL7614317 0.88 SLC2A1 (0.56) SLC2A1ACHETRPV1IMPDH2TP53
SCHEMBL7615766 0.88 SLC2A1 (0.56) SLC2A1ACHECA12CA9CA1
SCHEMBL7614313 0.88 SLC2A1 (0.56) SLC2A1ACHETRPV1IMPDH2TP53
SCHEMBL7621018 0.86 SLC2A1 (0.54) SLC2A1ACHECA12CA9CA1
SCHEMBL7621013 0.86 SLC2A1 (0.54) SLC2A1ACHECA12CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100495-A4 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORP (US) 2002-09-25 EP claimed
JP-2002521441-A 2002-07-16 JP claimed
EP-1100495-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP claimed
WO-2000006153-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO claimed
EP-1100495-A4 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORP (US) 2002-09-25 EP disclosed
EP-1100495-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP disclosed
WO-2000006153-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed