SCHEMBL7614435

SCHEMBL7614435

CCCCCCCOc1ccc(CCC(C)(N)CO)cc1OC

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 9/20 0.57
S1PR3 Q99500 7/20 0.49
S1PR4 O95977 6/20 0.49
S1PR5 Q9H228 5/20 0.49
KCNH2 Q12809 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
S1PR2 O95136 1/20 0.47
LPAR2 Q9HBW0 1/20 0.47
SPHK2 Q9NRA0 3/20 0.47
SPHK1 Q9NYA1 1/20 0.45
TNNC1 P63316 3/20 0.45
SGPL1 O95470 1/20 0.45
GPR183 P32249 1/20 0.45
CERS2 Q96G23 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8535469 0.89 S1PR1 (0.71) S1PR1S1PR3S1PR4S1PR5KCNH2
SCHEMBL12337601 0.87 S1PR1 (0.58) S1PR1S1PR3S1PR4S1PR5S1PR2
SCHEMBL7619599 0.87 S1PR1 (0.58) S1PR1S1PR3S1PR4S1PR5S1PR2
SCHEMBL3511041 0.86 ADRB2 (0.53) KCNH2TMEM97SIGMAR1
SCHEMBL3510320 0.86 ADRB2 (0.53) KCNH2TMEM97SIGMAR1
SCHEMBL2469791 0.84 S1PR1 (0.81) S1PR1S1PR3S1PR4S1PR5SPHK2
SCHEMBL2466810 0.84 S1PR1 (0.81) S1PR1S1PR3S1PR4S1PR5SPHK2
SCHEMBL2467762 0.84 S1PR1 (0.81) S1PR1S1PR3S1PR4S1PR5SPHK2
Hydrochloric Acid SCHEMBL2463923 0.83 S1PR1 (0.80) S1PR1S1PR3S1PR4S1PR5SPHK2
Hydrochloric Acid SCHEMBL2463212 0.83 S1PR1 (0.80) S1PR1S1PR3S1PR4S1PR5SPHK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778263-B1 BENZENE COMPOUND AND MEDICINAL USE THEREOF WELFIDE CORP (JP) 2002-01-09 EP claimed
US-5948820-A IMMUNOSUPPRESSANT; PREVENT REJECTION OF ORGAN TRANSPLANT;AUTOIMMUNE DISEASES; MULTIPLE SCLEROSIS; LUPUS; ANTIALLERGENS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-07 US claimed
EP-0778263-A1 BENZENE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-11 EP claimed
US-6372800-B1 IMMUNOSUPPRESSIVE EFFECT AND IS USEFUL AS AN INHIBITOR FOR THE REJECTION REACTION OCCURRING IN ORGAN OR BONE MARROW TRANSPLANTATION, AND AS A PREVENTIVE OR REMEDY FOR ARTICULAR RHEUMATISM, ATOPIC ECZEMA (DERMATITIS), BEHCET'S DISEASE, MITSUBISHI PHARMA CORPORATION (JP) 2002-04-16 US disclosed
EP-0778263-B1 BENZENE COMPOUND AND MEDICINAL USE THEREOF WELFIDE CORP (JP) 2002-01-09 EP disclosed
US-6187821-B1 SUCH AS 2-AMINO-2-(3-(4-HEPTYLPHENYL)PROPYL)BUTANE-1,4-DIOL; IMMUNOSUPPRESSANT; ADMINISTERING TO TREAT OR PREVENT AUTOIMMUNE DISEASES AND ALLERGIES WELFIDE CORPORATION (JP) 2001-02-13 US disclosed
US-5948820-A IMMUNOSUPPRESSANT; PREVENT REJECTION OF ORGAN TRANSPLANT;AUTOIMMUNE DISEASES; MULTIPLE SCLEROSIS; LUPUS; ANTIALLERGENS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-07 US disclosed
EP-0778263-A1 BENZENE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-11 EP disclosed