SCHEMBL7614849

SCHEMBL7614849

CCCCn1c(=O)c(NC(=O)Nc2c(C(C)C)ccc(N)c2C(C)C)c(-c2cccc(OC)c2)c2cccnc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ACAT1 P24752 1/20 0.70
SOAT1 P35610 3/20 0.68
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6638805 0.91 ACAT1 (0.75) ACAT1SOAT1KMT2A
SCHEMBL7615047 0.90 ACAT1 (0.85) ACAT1SOAT1
SCHEMBL6635737 0.89 ACAT1 (0.72) ACAT1SOAT1KMT2A
SCHEMBL7639342 0.89 ACAT1 (0.69) ACAT1SOAT1
SCHEMBL8328241 0.88 ACAT1 (0.71) ACAT1SOAT1KMT2A
SCHEMBL8328816 0.88 ACAT1 (0.71) ACAT1SOAT1KMT2A
SCHEMBL8328319 0.88 ACAT1 (0.71) ACAT1SOAT1KMT2A
SCHEMBL7613796 0.88 ACAT1 (0.74) ACAT1SOAT1KMT2A
SCHEMBL7614056 0.87 ACAT1 (0.74) ACAT1SOAT1KMT2A
SCHEMBL6635880 0.87 ACAT1 (0.68) ACAT1SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420381-B1 ACYL-COA: CHOLESTEROL ACYL TRANSFERASE (ACAT) INHIBITORY ACTIVITY, AND IS USEFUL AS AN AGENT FOR TREATMENT OF HYPERLIPIDEMIA AND ATHEROSCLEROSIS. SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2002-07-16 US disclosed
EP-1104763-A1 NAPHTHYRIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-06-06 EP disclosed