SCHEMBL7615401

SCHEMBL7615401

O=C(O)/C=C/c1ccc2c(c1)CCCC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.53
HSD17B10 Q99714 4/20 0.53
ALDH1A1 P00352 4/20 0.53
CA12 O43570 3/20 0.53
CA1 P00915 3/20 0.53
CA2 P00918 3/20 0.53
CA3 P07451 3/20 0.53
CA4 P22748 3/20 0.53
CA6 P23280 3/20 0.53
CA5A P35218 3/20 0.53
CA7 P43166 3/20 0.53
CA9 Q16790 3/20 0.53
CA14 Q9ULX7 3/20 0.53
CA5B Q9Y2D0 3/20 0.53
MAPK1 P28482 3/20 0.53
AKR1B10 O60218 2/20 0.53
AKR1B1 P15121 2/20 0.53
DPP4 P27487 2/20 0.53
HPGD P15428 2/20 0.53
HDAC3 O15379 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7615406 1.00 KDM4E (0.53) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL2728401 0.96 KDM4E (0.53) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL2728405 0.96 KDM4E (0.53) KDM4EHSD17B10ALDH1A1CA12CA1
Hydrochloric Acid SCHEMBL27910221 0.95 KDM4E (0.51) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL13797243 0.93 KDM4E (0.56) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL20681307 0.93 KDM4E (0.56) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL30207038 0.93 KDM4E (0.56) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL30567327 0.93 KDM4E (0.56) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL30263749 0.93 KDM4E (0.56) KDM4EHSD17B10ALDH1A1CA12CA1
SCHEMBL6264682 0.87 HSD17B10 (0.52) KDM4EHSD17B10ALDH1A1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100495-A4 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORP (US) 2002-09-25 EP disclosed
EP-1100495-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP disclosed
WO-2000006153-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed