SCHEMBL7618873

SCHEMBL7618873

Cc1cn2c(Cc3ccccc3)c(C3CC3)c(C(=O)C(N)=O)c2c(C(=O)C(=O)O)n1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PLA2G1B P04054 18/20 0.55
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
PLA2G2A P14555 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7643915 0.92 PLA2G1B (0.48) PLA2G1BPLA2G2A
SCHEMBL7189199 0.84 PLA2G1B (0.64) PLA2G1BPLA2G2A
SCHEMBL7645569 0.83 PLA2G1B (0.55) PLA2G1BPLA2G2A
SCHEMBL7185931 0.77 PLA2G1B (0.56) PLA2G1BPLA2G2A
SCHEMBL7621908 0.75 PLA2G1B (0.49) PLA2G1BPLA2G2A
SCHEMBL7616781 0.74 PLA2G1B (0.47) PLA2G1BPLA2G2A
SCHEMBL7641632 0.73 PLA2G1B (0.54) PLA2G1BPLA2G2A
SCHEMBL7647147 0.72 PLA2G1B (0.55) PLA2G1BPLA2G2A
SCHEMBL7643254 0.71 PLA2G1B (0.52) PLA2G1BPLA2G2A
SCHEMBL7015420 0.71 PLA2G1B (0.85) PLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265607-A2 METHOD FOR THE TREATMENT OF RENAL DYSFUNCTION WITH sPLA 2 INHIBITORS ELI LILLY AND COMPANY (US) 2002-12-18 EP disclosed
WO-2001066110-A2 METHOD FOR THE TREATMENT OF RENAL DYSFUNCTION WITH sPLA2 INHIBITORS ELI LILLY AND COMPANY (US) 2001-09-13 WO disclosed