SCHEMBL7619463

SCHEMBL7619463

COc1ccc(NC(=O)C=Cc2ccoc2)cc1OCCCN(C(C)C)C(C)C

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.59
BCHE P06276 14/20 0.49
ACHE P22303 13/20 0.49
TRPV1 Q8NER1 1/20 0.46
POLB P06746 2/20 0.45
GAA P10253 1/20 0.45
HTR2C P28335 1/20 0.44
MCHR1 Q99705 1/20 0.44
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7619454 1.00 SLC2A1 (0.59) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7606787 0.95 SLC2A1 (0.65) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7606790 0.95 SLC2A1 (0.65) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7606539 0.87 SLC2A1 (0.51) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7606541 0.87 SLC2A1 (0.51) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7619476 0.87 BCHE (0.54) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7614843 0.85 SLC2A1 (0.64) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7612941 0.85 SLC2A1 (0.66) SLC2A1BCHEACHETRPV1POLB
SCHEMBL7612346 0.85 SLC2A1 (0.56) SLC2A1BCHEACHEHTR2CMCHR1
SCHEMBL7620250 0.85 SLC2A1 (0.66) SLC2A1BCHEACHETRPV1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100495-A4 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORP (US) 2002-09-25 EP disclosed
EP-1100495-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP disclosed
WO-2000006153-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed