SCHEMBL7625286

SCHEMBL7625286

COC(=O)c1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCC3)cc1

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.82
CCR5 P51681 16/20 0.59
CXCR3 P49682 3/20 0.59
CCR7 P32248 2/20 0.59
CXCR5 P32302 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7624949 0.92 CCR2 (0.85) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL5204966 0.90 CCR2 (1.00) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7616230 0.90 CCR2 (0.74) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL5240554 0.88 CCR2 (0.82) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL5208811 0.87 CCR2 (0.81) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7958933 0.85 CCR2 (0.61) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL14032001 0.85 CCR2 (0.75) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7616237 0.84 CCR2 (0.77) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7216624 0.84 CCR2 (0.74) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL7222327 0.83 CCR2 (0.72) CCR2CCR5CXCR3CCR7CXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376536-B1 VIRICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-04-23 US disclosed
EP-1104416-A2 QUATERNARY AMMONIUM SALTS AND THEIR USE AS ANTI-HIV AGENTS Takeda Chemical Industries, Ltd. (JP) 2001-06-06 EP disclosed
US-6096780-A ANTIVIRAL COMPOUND USEFUL FOR TREATING HIV VIRUSES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-08-01 US disclosed
WO-2000010965-A2 QUATERNARY AMMONIUM SALTS AND THEIR USE AS ANTI-HIV AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-03-02 WO disclosed