SCHEMBL762669

SCHEMBL762669

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)c3cccc(OC)c3)C2)nc2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 7/20 0.48
KCNH2 Q12809 6/20 0.48
CYP2D6 P10635 3/20 0.48
CHRM1 P11229 1/20 0.48
CYP3A4 P08684 1/20 0.43
TP53 P04637 3/20 0.42
MAPT P10636 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762869 0.92 KCNH2 (0.48) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL742589 0.92 KCNH2 (0.48) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL762868 0.87 KCNH2 (0.45) HRH1KCNH2CYP2D6CHRM1SMN1; SMN2
SCHEMBL763828 0.86 KCNH2 (0.43) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL740346 0.86 HRH1 (0.47) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL740032 0.86 KCNH2 (0.48) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL740033 0.86 KCNH2 (0.48) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL762727 0.84 KCNH2 (0.51) HRH1KCNH2CYP2D6CHRM1USP2
SCHEMBL741653 0.84 L3MBTL1 (0.43) HRH1KCNH2CYP2D6CHRM1CYP3A4
SCHEMBL741655 0.84 L3MBTL1 (0.43) HRH1KCNH2CYP2D6CHRM1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed