SCHEMBL762969

SCHEMBL762969

CCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(N4CCC(O)CC4)cc3)C2)nc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 9/20 0.46
CYP2D6 P10635 7/20 0.46
KCNH2 Q12809 11/20 0.44
CHRM1 P11229 3/20 0.44
TP53 P04637 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CB P42338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762670 0.94 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL763356 0.93 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL762972 0.93 HRH1 (0.45) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL741823 0.92 HRH1 (0.44) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL741824 0.92 HRH1 (0.44) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL762802 0.92 HRH1 (0.43) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL763197 0.88 HRH1 (0.47) HRH1CYP2D6KCNH2CHRM1ALDH1A1
SCHEMBL763295 0.87 TP53 (0.44) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL741579 0.86 KCNH2 (0.45) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL741578 0.86 KCNH2 (0.45) HRH1CYP2D6KCNH2CHRM1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed