SCHEMBL7635650

SCHEMBL7635650

CC1(C)OC(=O)Nc2ncc(-c3cccc(Cl)c3)cc21

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.65
NR3C1 P04150 1/20 0.45
NR3C2 P08235 1/20 0.45
AR P10275 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3869106 0.79 PGR (1.00) PGRNR3C1NR3C2AR
SCHEMBL27558933 0.75 PGR (0.49) PGR
SCHEMBL14818906 0.72 PGR (0.39) PGRNR3C1NR3C2AR
SCHEMBL3379932 0.72 PGR (0.39) PGRNR3C1NR3C2AR
SCHEMBL7167921 0.71 PGR (0.60) PGRNR3C1NR3C2AR
SCHEMBL3380290 0.69 PGR (0.37) PGRNR3C1NR3C2AR
SCHEMBL3872465 0.68 PGR (0.82) PGRNR3C1NR3C2AR
SCHEMBL5125520 0.68 PGR (0.66) PGRNR3C1NR3C2AR
SCHEMBL3379455 0.68 NPC1 (0.44) PGRNR3C1NR3C2AR
SCHEMBL27579723 0.67 PGR (0.73) PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002543119-A 2002-12-17 JP claimed
JP-2002543206-A 2002-12-17 JP claimed
US-6399593-B1 CONTRACEPTIVES WYETH 2002-06-04 US claimed
US-6369056-B1 AGONISTS AND ANTAGONISTS OF THE PROGESTERONE RECEPTOR; CONTRACEPTIVES; 6-(3-CHLOROPHENYL)-4,4-DIMETHYL-1,4-DIHYDRO -3-OXA-1,8-DIAZA-NAPHTHALENE-2-ONE AND 6-CHLORO-4,4-DIMETHYL-1,4-DIHYDRO-3-OXA-1,5-DIAZA-NAPHTHALEN-2-ONE AMERICAN HOME PRODUCTS CORPORATION 2002-04-09 US claimed
EP-1173208-A2 CONTRACEPTIVE COMPOSITIONS CONTAINING CYCLIC UREA AND AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2002-01-23 EP claimed
EP-1173443-A1 CYCLIC UREA AND CYCLIC AMIDE DERIVATIVES American Home Products Corporation (US) 2002-01-23 EP claimed
WO-2000066103-A2 CONTRACEPTIVE COMPOSITIONS CONTAINING CYCLIC UREA AND AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO claimed
WO-2000066592-A1 CYCLIC UREA AND CYCLIC AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO claimed
US-20020111355-A1 Cyclic urea and cyclic amide derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 2002-08-15 US disclosed
US-6399593-B1 CONTRACEPTIVES WYETH 2002-06-04 US disclosed
US-6369056-B1 AGONISTS AND ANTAGONISTS OF THE PROGESTERONE RECEPTOR; CONTRACEPTIVES; 6-(3-CHLOROPHENYL)-4,4-DIMETHYL-1,4-DIHYDRO -3-OXA-1,8-DIAZA-NAPHTHALENE-2-ONE AND 6-CHLORO-4,4-DIMETHYL-1,4-DIHYDRO-3-OXA-1,5-DIAZA-NAPHTHALEN-2-ONE AMERICAN HOME PRODUCTS CORPORATION 2002-04-09 US disclosed
EP-1173208-A2 CONTRACEPTIVE COMPOSITIONS CONTAINING CYCLIC UREA AND AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2002-01-23 EP disclosed
EP-1173443-A1 CYCLIC UREA AND CYCLIC AMIDE DERIVATIVES American Home Products Corporation (US) 2002-01-23 EP disclosed
WO-2000066103-A2 CONTRACEPTIVE COMPOSITIONS CONTAINING CYCLIC UREA AND AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO disclosed
WO-2000066592-A1 CYCLIC UREA AND CYCLIC AMIDE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020111355-A1 Cyclic urea and cyclic amide derivatives PGR, GNRHR, FSHR PGR 1/4885NR3C1 41/4885NR3C2 36/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.