SCHEMBL7641995

SCHEMBL7641995

COC(=O)C(O)c1ccc(CCC(=O)O)c(NC(=O)OC(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 2/20 0.38
POLB P06746 1/20 0.36
BRD4 O60885 1/20 0.35
ACE P12821 1/20 0.34
BACE1 P56817 2/20 0.33
CPT1A P50416 1/20 0.33
CPT1B Q92523 1/20 0.33
HDAC1 Q13547 1/20 0.33
CNR2 P34972 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
SYK P43405 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4679329 0.83 SMN1; SMN2 (0.46) POLB
SCHEMBL6802648 0.76 LMNA (0.45) POLBBRD4ACECNR2ITGB1
SCHEMBL28809491 0.74 MAPT (0.35)
SCHEMBL5552326 0.74 NR1H2 (0.42) POLBBRD4ACEHDAC1CNR2
SCHEMBL26016215 0.73 CYP17A1 (0.46) PPARGPPARA
SCHEMBL6502501 0.71 LMNA (0.43) POLBBRD4HDAC1CNR2BRD9
SCHEMBL2349796 0.71 IDO1 (0.46) BRD4BACE1HDAC1PPARGSYK
SCHEMBL7217624 0.70 NQO2 (0.41) POLBBRD4HDAC1CNR2ITGB1
SCHEMBL28492620 0.68 NQO2 (0.41) POLBITGB1ITGA4
SCHEMBL10785428 0.68 SLC16A3 (0.43) POLBHDAC1CNR2BRD9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171113-A1 COMPOUNDS USEFUL AS PHOSPHOTYROSINE MIMICS Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-01-16 EP disclosed
WO-2000062770-A1 COMPOUNDS USEFUL AS PHOSPHOTYROSINE MIMICS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2000-10-26 WO disclosed
EP-1045836-A1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2000-10-25 EP disclosed
WO-1999031066-A1 PYRIDONES AS SRC FAMILY SH2 DOMAIN INHIBITORS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1999-06-24 WO disclosed