Acrylic Acid Methyl Ester

Acrylic Acid Methyl Ester

SCHEMBL7643475

Br.C=CC(=O)OC.CN(C)C

nearest known ligand 0.46

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Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Acrylic Acid Methyl Ester. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
TSHR P16473 9/20 0.38
HPGD P15428 1/20 0.37
ALDH1A1 P00352 10/20 0.36
TP53 P04637 3/20 0.36
HIF1A Q16665 3/20 0.36
CYP3A4 P08684 2/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.32
TGM2 P21980 1/20 0.31
THRB P10828 2/20 0.31
FGFR4 P22455 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acrylic Acid Methyl Ester SCHEMBL6932742 0.97 HCAR2 (0.48) HCAR2KEAP1NFE2L2TSHRHPGD
Acrylic Acid Methyl Ester SCHEMBL27465044 0.95 HCAR2 (0.46) HCAR2KEAP1NFE2L2TSHRHPGD
Acrylic Acid Methyl Ester SCHEMBL27696952 0.92 HCAR2 (0.43) HCAR2KEAP1NFE2L2TSHRHPGD
Acrylic Acid Methyl Ester SCHEMBL28476990 0.92 HCAR2 (0.43) HCAR2KEAP1NFE2L2TSHRHPGD
Acrylic Acid Methyl Ester SCHEMBL27524008 0.92 HCAR2 (0.43) HCAR2KEAP1NFE2L2TSHRHPGD
Acrylic Acid Methyl Ester SCHEMBL27897238 0.92
Acrylic Acid Methyl Ester SCHEMBL28087356 0.89
Acrylic Acid Methyl Ester SCHEMBL9108 0.89
Acrylic Acid Methyl Ester SCHEMBL7645157 0.89 HCAR2 (0.56) HCAR2KEAP1NFE2L2TSHRHPGD
Acrylic Acid Methyl Ester SCHEMBL1854813 0.89 HCAR2 (0.56) HCAR2KEAP1NFE2L2TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101879140-A The nanoparticle and the sustained release compositions that comprise aryl-heterocyclic compounds ELAN PHARMA INT LTD 2010-11-10 CN claimed
CN-101287451-A Nanoparticulate and controlled release compositions comprising a platelet aggregation inhibitor ELAN PHARMA INT LTD (IE) 2008-10-15 CN claimed
CN-101287453-A Nanoparticulate and controlled release compositions comprising a cephalosporin ELAN PHARMA INT LTD (IE) 2008-10-15 CN claimed
CN-101242813-A Nanoparticulate and controlled release compositions comprising aryl-heterocyclic compounds ELAN PHARMA INT LTD (IE) 2008-08-13 CN claimed
US-6482875-B2 ORGANIC FIBROUS MATERIAL AND A BINDER CONTAINING AT LEAST TWO DIFFERENT POLYACRYLATES; COMPOSITE HAS A FLOW TRANSITION RANGE OF 70 DEGREES C. TO 130 DEGREES C. DORUS KLEBETECHNIK GMBH & CO. KG (DE) 2002-11-19 US disclosed
US-20020032253-A1 Organic fibrous material and a binder containing at least two different polyacrylates; composite has a flow transition range of 70 degrees C. to 130 degrees C. HENKEL DORUS GMBH & CO. KG (DE) 2002-03-14 US disclosed