SCHEMBL7643596

SCHEMBL7643596

NC(Cc1ccccc1)C(=O)NCCc1c[nH]cn1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
NLN Q9BYT8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7645866 1.00 KMT2A (0.45) KMT2ACA12CA1CA2NLN
SCHEMBL7643594 1.00 KMT2A (0.45) KMT2ACA12CA1CA2NLN
Bromide SCHEMBL9551371 0.99 KMT2A (0.44) KMT2ACA12CA1CA2NLN
SCHEMBL7618103 0.91 LTA4H (0.48)
SCHEMBL7618099 0.91 LTA4H (0.48)
SCHEMBL23573011 0.90 NLN (0.47) NLN
SCHEMBL13073718 0.90 NLN (0.47) NLN
SCHEMBL21794913 0.90 NLN (0.47) NLN
SCHEMBL7622435 0.89 CTSC (0.42)
SCHEMBL3217867 0.89 CTSC (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448282-B1 H3 HISTAMINE RECEPTOR ANTAGONIST ACTIVITY; ALLERGY, INFLAMMATION, CARDIOVASCULAR DISEASE, DEPRESSION, SCHIZOPHRENIA, NARCOLEPSY, SLEEP APNEA, INSOMNIA, EPILEPSY, HYPOTHALAMIC DYSFUNCTION GLIATECH, INC. 2002-09-10 US disclosed
US-6166060-A 1H-4(5)-substituted imidazole derivatives GLIATECH, INC. (US) 2000-12-26 US disclosed