SCHEMBL7644374

SCHEMBL7644374

COC(=O)c1cc(/C=C/c2cccc(F)c2)ccc1NC(=O)c1ccc(N(C)C(=O)c2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
KDM4E B2RXH2 3/20 0.41
SNCA P37840 3/20 0.39
APP P05067 1/20 0.39
SMN1; SMN2 Q16637 6/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KCNK2 O95069 1/20 0.38
POLB P06746 3/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7644381 1.00 CYP1A2 (0.43) CYP1A2CYP2C19CYP2D6TSHRNPC1
SCHEMBL7534688 0.95 TSHR (0.45) CYP1A2CYP2C19CYP2D6TSHRNPC1
SCHEMBL7534682 0.95 TSHR (0.45) CYP1A2CYP2C19CYP2D6TSHRNPC1
SCHEMBL7650286 0.92 CYP1A2 (0.48) CYP1A2CYP2C19CYP2D6TSHRNPC1
SCHEMBL7650281 0.92 CYP1A2 (0.48) CYP1A2CYP2C19CYP2D6TSHRNPC1
SCHEMBL7648625 0.92 APP (0.46) CYP1A2CYP2C19CYP2D6TSHRKDM4E
SCHEMBL7648628 0.92 APP (0.46) CYP1A2CYP2C19CYP2D6TSHRKDM4E
SCHEMBL7645168 0.88 SNCA (0.46) CYP1A2CYP2C19CYP2D6TSHRKDM4E
SCHEMBL7529853 0.87 APP (0.47) CYP1A2CYP2C19CYP2D6TSHRKDM4E
SCHEMBL7529846 0.87 APP (0.47) CYP1A2CYP2C19CYP2D6TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479548-B2 P-(BENZOYLAMINO)STILBENE DERIVATIVES TELIK, INC. 2002-11-12 US disclosed