SCHEMBL7646263

SCHEMBL7646263

Fc1ccc(-c2[nH]c3ccccc3c2CCN2CCCCC2)cc1

nearest known ligand 0.81

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 10/20 0.81
HTR2C P28335 9/20 0.81
DRD2 P14416 8/20 0.81
CHRNA7 P36544 1/20 0.45
APOL1 O14791 1/20 0.44
KCNH2 Q12809 2/20 0.44
MPO P05164 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524422 0.89 HTR2A (1.00) HTR2AHTR2CDRD2CHRNA7KCNH2
SCHEMBL7645809 0.89 HTR2A (1.00) HTR2AHTR2CDRD2CHRNA7KCNH2
SCHEMBL7648046 0.88 HTR2A (1.00) HTR2AHTR2CDRD2KCNH2
SCHEMBL7649978 0.86 HTR2A (0.75) HTR2AHTR2CDRD2KCNH2MPO
SCHEMBL7649032 0.86 HTR2A (0.75) HTR2AHTR2CDRD2MPO
SCHEMBL10832307 0.82 HTR2A (0.73) HTR2AHTR2CDRD2CHRNA7MPO
SCHEMBL7646650 0.81 HTR2A (0.79) HTR2AHTR2CDRD2KCNH2
SCHEMBL10832216 0.81 HTR2A (0.72) HTR2AHTR2CDRD2CHRNA7
SCHEMBL25772732 0.78 HTR2A (0.68) HTR2AHTR2CDRD2CHRNA7KCNH2
SCHEMBL7646923 0.78 HTR2A (0.69) HTR2AHTR2CDRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999011619-A1 PHENYLINDOLE DERIVATIVES AS 5-HT2A RECEPTOR LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1999-03-11 WO claimed
US-6486153-B1 Phenylindole derivatives as 5-HT2A receptor ligands MERCK SHARP & DOHME LTD. 2002-11-26 US disclosed
WO-1999011619-A1 PHENYLINDOLE DERIVATIVES AS 5-HT2A RECEPTOR LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1999-03-11 WO disclosed