SCHEMBL7646709

SCHEMBL7646709

C=CCC(=O)OC1c2ccccc2-c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
NPSR1 Q6W5P4 1/20 0.38
CYP2D6 P10635 2/20 0.37
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 2/20 0.35
TSHR P16473 2/20 0.35
MAPT P10636 1/20 0.34
HTT P42858 2/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21778843 0.81 POLB (0.46) POLBCYP2D6HDAC3HDAC4HDAC7
SCHEMBL27555134 0.80 POLB (0.48) POLBCYP2D6HDAC3HDAC4HDAC7
SCHEMBL21758220 0.78 POLB (0.43) POLBCYP2D6HDAC3HDAC4HDAC7
SCHEMBL240153 0.77 POLB (0.46) POLBALDH1A1GAAHDAC3HDAC4
SCHEMBL27593730 0.77 POLB (0.46) POLBCYP2D6ALDH1A1HDAC3HDAC4
SCHEMBL31390251 0.77 POLB (0.46) POLBALDH1A1GAAHDAC3HDAC4
SCHEMBL3754584 0.77 POLB (0.50) POLBCYP2D6GAAHDAC3HDAC4
SCHEMBL17995090 0.76 MAPT (0.38) POLBALDH1A1TSHRMAPTKMT2A
SCHEMBL27864062 0.75 POLB (0.47) POLBNPSR1ALDH1A1HDAC3HDAC4
SCHEMBL6910125 0.75 POLB (0.43) POLBALDH1A1GAAHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6458760-B1 COMPRISING ADMINISTERING TO SAID PATIENT A THERAPEUTICALLY EFFECTIVE AMOUNT OF A COMPOUND WHICH IS A SPECIFIC INHIBITOR OF EITHER CATHEPSIN B OR CATHEPSIN L, BUT WHICH IS NOT AS EFFECTIVE INHIBITOR OF CALPAIN HENRY FORD HEALTH SYSTEM 2002-10-01 US disclosed