SCHEMBL7647490

SCHEMBL7647490

CCc1cccc(N(C)C(N)=Nc2ccc(I)cc2)c1

nearest known ligand 0.78

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 0.78
TP53 P04637 1/20 0.59
CYP2D6 P10635 1/20 0.59
TSHR P16473 1/20 0.59
THPO P40225 1/20 0.59
MTOR P42345 1/20 0.59
MEN1 O00255 1/20 0.58
LMNA P02545 1/20 0.58
MAPT P10636 1/20 0.58
PMP22 Q01453 1/20 0.58
KMT2A Q03164 1/20 0.58
TDP1 Q9NUW8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6158218 0.86 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7642451 0.86 SIGMAR1 (0.60) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7641508 0.83 SIGMAR1 (0.53) SIGMAR1
SCHEMBL6727463 0.82 SIGMAR1 (0.85) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6719522 0.81 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6720812 0.79 SIGMAR1 (0.85) SIGMAR1
SCHEMBL6724568 0.78 SIGMAR1 (0.77) SIGMAR1
SCHEMBL8194426 0.77 SIGMAR1 (0.75) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL8497150 0.77 SIGMAR1 (0.75) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6717192 0.76 SIGMAR1 (0.73) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0517852-B1 TRI- AND TETRA-SUBSTITUTED GUANIDINES AND THEIR USE AS EXCITATORY AMINO ACID ANTAGONISTS OREGON STATE (US) 2002-07-10 EP claimed