SCHEMBL7651020

SCHEMBL7651020

CCC(N)OC(=O)/C=C/C(=O)OC(N)CC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 9/20 0.41
ATM Q13315 1/20 0.37
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
GFPT1 Q06210 1/20 0.35
TSHR P16473 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SLC1A3 P43003 1/20 0.31
SLC1A2 P43004 1/20 0.31
SLC1A1 P43005 1/20 0.31
LAP3 P28838 1/20 0.31
GABRP O00591 2/20 0.30
GABRD O14764 2/20 0.30
GABRA1 P14867 2/20 0.30
GABRB1 P18505 2/20 0.30
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30
GABRA5 P31644 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878831 1.00 HCAR2 (0.41) HCAR2ATMKEAP1NFE2L2GFPT1
SCHEMBL2388631 0.82 GFPT1 (0.43) HCAR2ATMGFPT1MAPTRAB9A
SCHEMBL27991557 0.82 HCAR2 (0.39) HCAR2ATMKEAP1NFE2L2GFPT1
SCHEMBL4353141 0.82 HCAR2 (0.39) HCAR2ATMKEAP1NFE2L2GFPT1
SCHEMBL149786 0.82
Bromide SCHEMBL29244222 0.80 TSHR (0.41) TSHRLAP3
Hydrochloric Acid SCHEMBL28480383 0.80 TSHR (0.41) TSHRLAP3
SCHEMBL28180758 0.79 ATM (0.45) HCAR2ATMTSHRMAPTRAB9A
Butane SCHEMBL1034123 0.79 TSHR (0.42) TSHRLAP3
SCHEMBL2110683 0.77 TSHR (0.35) TSHRSLC1A3SLC1A2SLC1A1LAP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1235870-C Novel use of phenyl hetero alkylamine derivatives ASTRAZENECA AB (SE) 2006-01-11 CN disclosed
CN-1411435-A Novel use of phenylheteroalkylamine derivatives ASTRAZENECA AB (SE) 2003-04-16 CN disclosed
US-6479534-B1 Indoline derivatives and method of treating obesity VERNALIS RESEARCH LIMITED (GB) 2002-11-12 US disclosed