SCHEMBL7651189

SCHEMBL7651189

COc1ccccc1CNC(=O)c1ccccc1N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 12/20 1.00
ALDH1A1 P00352 8/20 1.00
KDM4E B2RXH2 5/20 1.00
RCE1 Q9Y256 1/20 1.00
HTT P42858 2/20 0.64
GAA P10253 2/20 0.64
PKM P14618 1/20 0.64
KMT2A Q03164 1/20 0.63
NPC1 O15118 1/20 0.62
HDAC1 Q13547 1/20 0.60
PLA2G1B P04054 1/20 0.60
ATG4B Q9Y4P1 1/20 0.60
NLRP3 Q96P20 1/20 0.60
USP2 O75604 1/20 0.59
TDP1 Q9NUW8 1/20 0.58
TP53 P04637 1/20 0.57
GLA P06280 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28478696 0.86 HPGD (0.76) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL19326905 0.85 HPGD (0.74) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL29508722 0.85 HPGD (0.79) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL5597952 0.84 HPGD (0.73) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL19747579 0.83 HPGD (0.78) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL28729043 0.81 HPGD (1.00) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL3208233 0.81 HPGD (0.67) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL27463741 0.81 HPGD (0.79) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL6005231 0.80 HPGD (0.66) HPGDALDH1A1KDM4ERCE1HTT
SCHEMBL22972357 0.80 HPGD (0.72) HPGDALDH1A1KDM4ERCE1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed