SCHEMBL7651344

SCHEMBL7651344

CCOC(=O)CCSc1ccc(Br)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.51
KCNH2 Q12809 1/20 0.51
ALDH1A1 P00352 6/20 0.49
PKM P14618 1/20 0.49
HTT P42858 1/20 0.49
MAPT P10636 6/20 0.48
SDCBP O00560 1/20 0.48
SDC2 P34741 1/20 0.48
KMT2A Q03164 3/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
MEN1 O00255 1/20 0.46
S1PR4 O95977 1/20 0.46
LMNA P02545 1/20 0.46
S1PR1 P21453 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15228885 0.91 SMN1; SMN2 (0.47) HSP90AA1KCNH2ALDH1A1MAPTSDCBP
SCHEMBL16334378 0.89 ALDH1A1 (0.46) HSP90AA1KCNH2ALDH1A1MAPTSDCBP
SCHEMBL13948873 0.87 ALDH1A1 (0.61) ALDH1A1PKMHTTMAPTKMT2A
SCHEMBL25270599 0.84 MAPT (0.55) ALDH1A1PKMHTTMAPTKMT2A
SCHEMBL28932704 0.84 HTT (0.68) ALDH1A1PKMHTTMAPTSDCBP
SCHEMBL11539971 0.83 SMN1; SMN2 (0.56) ALDH1A1MAPTKMT2AHPGDSMN1; SMN2
SCHEMBL7344673 0.83 ALDH1A1 (0.61) ALDH1A1MAPTKMT2AHPGDSMN1; SMN2
SCHEMBL7012446 0.83 HSP90AA1 (0.54) HSP90AA1KCNH2ALDH1A1PKMHTT
SCHEMBL6928975 0.83 ATM (0.57) ALDH1A1PKMHTTMAPTHPGD
SCHEMBL5450459 0.82 MAPT (0.47) ALDH1A1MAPTKMT2AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344463-B1 SKIN DISORDERS, ACNE ALLERGAN SALES, INC. 2002-02-05 US disclosed
EP-0636127-B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN INC (US) 2001-04-04 EP disclosed
US-6090826-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN SALES, INC. (US) 2000-07-18 US disclosed
US-5750693-A THIOCHROMANYL OR CHROMANYL COMPOUNDS AS ANTICARCINOGINIC AGENTS, SKIN DISORDERS AND ATHEROSCLEROSIS ALLERGAN (US) 1998-05-12 US disclosed
US-5677451-A CONTROLLING CELL DIFFERENTIATION; SKIN DISORDERS; ANTICANCER AGENTS ALLERGAN (US) 1997-10-14 US disclosed
US-5663347-A REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION; TREATMENT OF SKIN DISORDERS; ANTICARCINOGNIC AGENTS ALLERGAN (US) 1997-09-02 US disclosed
US-5468879-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1995-11-21 US disclosed
EP-0636127-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1995-02-01 EP disclosed
US-5264578-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1993-11-23 US disclosed
WO-1993016068-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1993-08-19 WO disclosed