SCHEMBL7651586

SCHEMBL7651586

CCC1(CC)CCOc2ccc(C#Cc3cnc(CCCCC(=O)O)cn3)cc21

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 16/20 0.37
CYP3A4 P08684 2/20 0.35
RARA P10276 1/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
KMT2A Q03164 1/20 0.35
PPARA Q07869 1/20 0.33
CYP26A1 O43174 1/20 0.33
FFAR1 O14842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8846432 0.90 CYP3A4 (0.40) PTGER4CYP3A4RARARARBRARG
SCHEMBL7654881 0.88 RARA (0.37) PTGER4CYP3A4RARARARBRARG
SCHEMBL8659621 0.81 CYP3A4 (0.42) CYP3A4RARARARBRARGKMT2A
SCHEMBL6684655 0.80 RARA (0.46) PTGER4CYP3A4RARARARBRARG
SCHEMBL8898602 0.79 POLB (0.38) PTGER4FFAR1
SCHEMBL7650441 0.79 CYP3A4 (0.41) CYP3A4RARARARBRARGKMT2A
SCHEMBL8875912 0.79 CYP3A4 (0.36) CYP3A4RARARARBRARGKMT2A
SCHEMBL7656133 0.78 CYP3A4 (0.39) PTGER4CYP3A4RARARARBRARG
SCHEMBL9673782 0.78 CYP3A4 (0.39) PTGER4CYP3A4RARARARBRARG
SCHEMBL7654875 0.78 CYP3A4 (0.43) PTGER4CYP3A4RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344463-B1 SKIN DISORDERS, ACNE ALLERGAN SALES, INC. 2002-02-05 US disclosed
EP-0636127-B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN INC (US) 2001-04-04 EP disclosed
US-6090826-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN SALES, INC. (US) 2000-07-18 US disclosed
US-5663347-A REGULATORS OF CELL PROLIFERATION AND DIFFERENTIATION; TREATMENT OF SKIN DISORDERS; ANTICARCINOGNIC AGENTS ALLERGAN (US) 1997-09-02 US disclosed
US-5468879-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1995-11-21 US disclosed
EP-0636127-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1995-02-01 EP disclosed
US-5264578-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN, INC. (US) 1993-11-23 US disclosed
WO-1993016068-A1 DISUBSTITUTED ACETYLENES BEARING HETEROBICYCLIC GROUPS AND HETEROAROMATIC OR PHENYL GROUPS HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC. (US) 1993-08-19 WO disclosed