SCHEMBL7651693

SCHEMBL7651693

CC[C@H](N)C(=O)N1c2cc3ccccc3cc2C[C@H]1C(=O)NCC(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
LMNA P02545 4/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5563790 0.96 KDM4E (0.53) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL5563791 0.96 KDM4E (0.53) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568891 0.86 KDM4E (0.51) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568561 0.83 KDM4E (0.39) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL5569402 0.83 KDM4E (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568302 0.77 KDM4E (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL7659015 0.77 KDM4E (0.48) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568546 0.76 KDM4E (0.80) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL6274286 0.76 KDM4E (0.80) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL7042292 0.76 KDM4E (0.80) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6335360-B1 INDOLINE-2-CARBOXYLIC AMIDE DERIVATIVES; OBESITY, EATING AND PSYCHOLOGICAL DISORDERS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-01-01 US disclosed