SCHEMBL5568561

SCHEMBL5568561

CC[C@H](NC(=O)OC(C)(C)C)C(=O)N1c2cc3ccccc3cc2C[C@H]1C(=O)NCC(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CXCR3 P49682 8/20 0.39
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
SCN9A Q15858 3/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5563327 0.88 CXCR3 (0.35) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5563179 0.87 KDM4E (0.37) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568446 0.86 ACE (0.42) CTSBCTSSCTSK
SCHEMBL5563142 0.86 GHSR (0.43) CXCR3SCN9AKMT2ALMNAPOLB
SCHEMBL5564142 0.86 CTSK (0.39) CTSBCTSSCTSKSCN9AKMT2A
SCHEMBL5564139 0.86 CTSK (0.39) CTSBCTSSCTSKSCN9AKMT2A
SCHEMBL7651693 0.83 KDM4E (0.56) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL5563790 0.81 KDM4E (0.53) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL5563791 0.81 KDM4E (0.53) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568286 0.80 CTSK (0.34) KDM4EALDH1A1CXCR3CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042288-B1 TRIPEPTIDYL PEPTIDASE INHIBITORS INST NAT SANTE RECH MED (FR) 2007-11-07 EP disclosed
US-6335360-B1 INDOLINE-2-CARBOXYLIC AMIDE DERIVATIVES; OBESITY, EATING AND PSYCHOLOGICAL DISORDERS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-01-01 US disclosed