SCHEMBL7652044

SCHEMBL7652044

O=c1c2ccccc2n(CCCCN2CCC(OC(c3ccccc3)c3ccccc3)CC2)c(=O)n1CCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 2/20 0.53
CACNA1H O95180 2/20 0.53
BCHE P06276 9/20 0.50
LMNA P02545 2/20 0.48
MEN1 O00255 1/20 0.48
UBE2N P61088 1/20 0.48
KMT2A Q03164 1/20 0.48
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HPGDS O60760 1/20 0.47
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
THRB P10828 1/20 0.44
NPC1 O15118 1/20 0.44
MLNR O43193 1/20 0.44
NR1I2 O75469 1/20 0.44
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
FYN P06241 1/20 0.44
CHRM2 P08172 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7651171 0.96 CACNA1G (0.53) CACNA1GCACNA1HBCHELMNAMEN1
Hydrochloric Acid SCHEMBL7650323 0.91 UBE2N (0.51) CACNA1GCACNA1HBCHELMNAMEN1
SCHEMBL7652346 0.90 BCHE (0.52) CACNA1GCACNA1HBCHELMNAMEN1
SCHEMBL7649679 0.89 BCHE (0.53) BCHELMNAMEN1UBE2NKMT2A
SCHEMBL7650486 0.89 BCHE (0.53) BCHELMNAMEN1UBE2NKMT2A
SCHEMBL7650856 0.89 BCHE (0.53) BCHELMNAMEN1UBE2NKMT2A
SCHEMBL7654660 0.89 BCHE (0.48) CACNA1GCACNA1HBCHELMNAMEN1
SCHEMBL7655637 0.89 BCHE (0.53) BCHELMNAMEN1UBE2NKMT2A
SCHEMBL7655890 0.89 BCHE (0.53) BCHELMNAMEN1UBE2NKMT2A
SCHEMBL7655620 0.88 BCHE (0.52) BCHELMNAMEN1UBE2NKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed