SCHEMBL7652491

SCHEMBL7652491

COC(=O)c1cc(C(C)(C)C(=O)OC)ccc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.54
ALDH1A1 P00352 5/20 0.54
GAA P10253 5/20 0.54
HSD17B10 Q99714 3/20 0.54
MAPT P10636 2/20 0.54
HPGD P15428 2/20 0.54
TSHR P16473 2/20 0.54
ALOX15 P16050 1/20 0.54
CFTR P13569 5/20 0.51
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
GLA P06280 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
ATM Q13315 1/20 0.45
ABL1 P00519 1/20 0.44
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA9 Q16790 3/20 0.37
CA5A P35218 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054575 0.85 ALDH1A1 (0.58) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL30033368 0.84 ALDH1A1 (0.57) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL31357589 0.81 CNR2 (0.60) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL1139411 0.81 CFTR (0.77) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL23582257 0.81 CNR2 (0.60) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL13264181 0.80 CNR1 (0.46) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL15456896 0.79 ALDH1A1 (0.50) KDM4EALDH1A1HSD17B10MAPTTSHR
SCHEMBL9612065 0.79 CNR1 (0.48) KDM4EALDH1A1GAAHSD17B10HPGD
SCHEMBL31292480 0.79 CNR2 (0.48) KDM4EALDH1A1GAAHSD17B10MAPT
SCHEMBL3445900 0.79 CNR1 (0.48) ALDH1A1CFTRCNR1CNR2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed