SCHEMBL7652512

SCHEMBL7652512

CCOC(=O)C(Oc1nc(C)cc(C)n1)C(=O)OCC

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.49
EDNRB P24530 4/20 0.41
EDNRA P25101 4/20 0.41
POLB P06746 2/20 0.41
NR1I2 O75469 1/20 0.41
KCNE1 P15382 1/20 0.41
KCNQ1 P51787 1/20 0.41
GAA P10253 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 4/20 0.41
MEN1 O00255 2/20 0.41
RAB9A P51151 2/20 0.41
THRB P10828 1/20 0.41
ALDH1A1 P00352 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9460647 0.83 HTT (0.47) HTTEDNRBEDNRAPOLBNR1I2
SCHEMBL7651729 0.79 EDNRB (0.51) EDNRBEDNRAPOLBNR1I2KCNE1
SCHEMBL9723575 0.77 EDNRB (0.47) HTTEDNRBEDNRAPOLBNR1I2
SCHEMBL7652517 0.74 HTT (0.51) HTTPOLBGAANPSR1KMT2A
SCHEMBL9460361 0.72 TDP1 (0.45) HTTEDNRBEDNRAPOLBNR1I2
SCHEMBL9357252 0.71 SMN1; SMN2 (0.49) EDNRBEDNRAPOLBNR1I2KCNE1
SCHEMBL9460319 0.71 TSHR (0.54) POLBGAANPSR1KMT2AMEN1
SCHEMBL15998733 0.71 EDNRB (0.56) EDNRBEDNRAPOLBNR1I2KCNE1
SCHEMBL9357632 0.70 EDNRB (0.50) EDNRBEDNRAPOLBNR1I2KCNE1
SCHEMBL28376192 0.70 HTT (0.47) HTTPOLBGAANPSR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6482947-B1 Substituted (hetero) aryl compounds, process for their preparation, agents containing them and their use as safeners HOECHST AKTIENGESELLSCHAFT (DE) 2002-11-19 US claimed