SCHEMBL7652987

SCHEMBL7652987

CC(=O)Nc1ccc(C#N)c2c1C(=O)C(=NO)CC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
HTT P42858 1/20 0.36
MAOA P21397 1/20 0.35
CASP3 P42574 1/20 0.33
KDM4E B2RXH2 3/20 0.32
HPGD P15428 3/20 0.32
GAA P10253 3/20 0.32
HSD17B10 Q99714 1/20 0.32
AR P10275 1/20 0.31
NOTUM Q6P988 1/20 0.31
PLA2G7 Q13093 1/20 0.31
MAPT P10636 2/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
NEU3 Q9UQ49 1/20 0.30
CXCR2 P25025 1/20 0.30
CCNE2 O96020 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653044 0.83 MAOA (0.38) ALDH1A1HTTMAOACASP3KDM4E
SCHEMBL7655842 0.82 CA1 (0.38) ALDH1A1MAOACASP3KDM4EHPGD
SCHEMBL7658801 0.82 KMT2A (0.39) ALDH1A1MAOACASP3KDM4EHPGD
SCHEMBL7654012 0.76 MAPT (0.41) ALDH1A1HTTMAOACASP3KDM4E
SCHEMBL7653367 0.74 MAOA (0.48) ALDH1A1MAOACASP3KDM4EHPGD
SCHEMBL24728326 0.73 CA1 (0.35) MAOAMEN1KMT2A
SCHEMBL26276091 0.72 CA1 (0.34) MAOA
SCHEMBL30977209 0.72 MEN1 (0.34) ALDH1A1MAOAKDM4EHSD17B10MAPT
SCHEMBL31421946 0.72 HDAC1 (0.34) ALDH1A1HTT
SCHEMBL27218964 0.72 MEN1 (0.34) MAOACASP3KDM4EHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407115-B1 ANTICARCINOGENIC AND ANTITUMOR AGENTS; SIDE EFFECT REDUCTION, WATER SOLUBILITY DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2002-06-18 US disclosed
US-5834476-A DERIVATIVE OF CAMPTOTHECIN, ANTITUMOR AGENT, ANTICARCINOGENIC AGENT DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-11-10 US disclosed
US-5770605-A Method for treating leukemia with a hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-06-23 US disclosed
US-5658920-A ANTITUMOR AGENTS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-08-19 US disclosed
US-5637770-A Hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-06-10 US disclosed
EP-0495432-B1 Hexa-cyclic compound DAIICHI SEIYAKU CO (JP) 1996-05-29 EP disclosed
EP-0495432-A1 Hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1992-07-22 EP disclosed