SCHEMBL7654426

SCHEMBL7654426

Brc1ccc2c(c1)c1cc(Br)ccc1n2C(CNCc1ccccc1)CN1CCNCC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BAX Q07812 2/20 0.50
MAPT P10636 2/20 0.49
CYP3A4 P08684 2/20 0.49
TP53 P04637 1/20 0.49
ALOX15 P16050 1/20 0.49
MAPK1 P28482 1/20 0.49
DNM1 Q05193 7/20 0.43
CXCR4 P61073 1/20 0.41
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
KMT2A Q03164 2/20 0.38
RAD52 P43351 2/20 0.38
MEN1 O00255 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL607992 0.77 BAX (0.60) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL5024339 0.69 BAX (0.72) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL29398838 0.69 BAX (0.72) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL607745 0.69 BAX (0.72) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL5024320 0.69 BAX (0.72) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL29992291 0.69 BAX (0.72) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL22261901 0.69 BAX (0.64) BAXMAPTCYP3A4TP53ALOX15
Hydrochloric Acid SCHEMBL31038642 0.69 MAPT (0.73) BAXMAPTCYP3A4TP53ALOX15
Hydrochloric Acid SCHEMBL29462932 0.69 MAPT (0.73) BAXMAPTCYP3A4TP53ALOX15
SCHEMBL608294 0.68 BAX (0.88) BAXMAPTCYP3A4TP53ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237887-A1 9-(PIPERAZINYLALKYL)CARBAZOLES AS BAX-MODULATORS Applied Research Systems ARS Holding N.V. (AN) 2002-09-11 EP claimed
WO-2001029028-A1 9- (PIPERAZINYLALKYL) CARBAZOLES AS BAX-MODULATORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-04-26 WO claimed