SCHEMBL7654430

SCHEMBL7654430

CCOC(=O)CCCCCn1c(=O)c2ccccc2n(CCCCBr)c1=O

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TNF P01375 6/20 0.70
CTNNB1 P35222 1/20 0.51
CNR2 P34972 5/20 0.49
ALDH1A1 P00352 3/20 0.49
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.47
TP53 P04637 1/20 0.47
PSEN1 P49768 1/20 0.47
PSEN2 P49810 1/20 0.47
APH1B Q8WW43 1/20 0.47
NCSTN Q92542 1/20 0.47
APH1A Q96BI3 1/20 0.47
PSENEN Q9NZ42 1/20 0.47
HDAC1 Q13547 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649768 1.00 TNF (0.70) TNFCTNNB1CNR2ALDH1A1HTT
SCHEMBL7649846 0.87 TNF (0.59) TNFCTNNB1CNR2ALDH1A1HTT
SCHEMBL7650022 0.87 TNF (0.73) TNFCTNNB1CNR2ALDH1A1TP53
SCHEMBL7648268 0.85 TNF (0.53) TNF
SCHEMBL7656518 0.84 TNF (0.67) TNFCTNNB1CNR2ALDH1A1HTT
SCHEMBL7648315 0.84 TNF (0.50) TNFALDH1A1KDM4E
SCHEMBL7651102 0.84 TNF (0.52) TNFCTNNB1ALDH1A1HDAC1
SCHEMBL1004476 0.83 TNF (0.63) TNFCTNNB1CNR2ALDH1A1HTT
SCHEMBL1004093 0.83 TNF (0.63) TNFCTNNB1CNR2ALDH1A1HTT
SCHEMBL7650027 0.83 TNF (0.68) TNFCTNNB1CNR2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed