SCHEMBL7654911

SCHEMBL7654911

CCOC(=O)C(C/C=C/c1ccccc1)C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
MMP8 P22894 2/20 0.50
CTDSP1 Q9GZU7 1/20 0.49
HTR2A P28223 3/20 0.49
TDP1 Q9NUW8 1/20 0.48
PAM P19021 1/20 0.47
RAB9A P51151 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GRIK1 P39086 2/20 0.47
GRIK2 Q13002 2/20 0.47
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
GLA P06280 1/20 0.46
PPARG P37231 1/20 0.46
ADORA3 P0DMS8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654904 1.00 MEN1 (0.50) MEN1KMT2AMMP8CTDSP1HTR2A
SCHEMBL7490894 0.95 GRIK1 (0.49) MEN1KMT2AMMP8CTDSP1HTR2A
SCHEMBL9620462 0.92 MMP8 (0.50) MEN1KMT2AMMP8CTDSP1HTR2A
SCHEMBL9620464 0.92 MMP8 (0.50) MEN1KMT2AMMP8CTDSP1HTR2A
SCHEMBL28952721 0.90 MEN1 (0.46) MEN1KMT2AMMP8CTDSP1HTR2A
SCHEMBL12123422 0.85 HTR2A (0.50) KMT2AHTR2ATDP1PAMGRIK1
SCHEMBL27629744 0.84 TDP1 (0.52) MEN1KMT2AMMP8CTDSP1TDP1
SCHEMBL7309863 0.84 GRIK1 (0.55) MEN1KMT2ACTDSP1HTR2APAM
Hydrochloric Acid SCHEMBL7309854 0.83 GRIK1 (0.54) MEN1KMT2ACTDSP1HTR2APAM
Hydrochloric Acid SCHEMBL7309856 0.83 GRIK1 (0.54) MEN1KMT2ACTDSP1HTR2APAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102875278-B Method for synthesizing optically-active 2-(2', 3'-allene group) malonate UNIV ZHEJIANG 2014-07-30 CN claimed
CN-102875278-A Method for synthesizing optically-active 2-(2', 3'-allene group) malonate UNIV ZHEJIANG 2013-01-16 CN claimed
CN-114890881-B Method for simply synthesizing allyl dicarbonyl compound 南阳师范学院 2023-06-02 CN disclosed
CN-114890881-A Method for simply synthesizing allyl dicarbonyl compound 南阳师范学院 2022-08-12 CN disclosed
CN-102875278-B Method for synthesizing optically-active 2-(2', 3'-allene group) malonate UNIV ZHEJIANG 2014-07-30 CN disclosed
CN-102875278-A Method for synthesizing optically-active 2-(2', 3'-allene group) malonate UNIV ZHEJIANG 2013-01-16 CN disclosed
US-6495370-B1 A METHOD FOR DETECTING A GLUTATHIONE-S-TRANSFERASE ISOENZYME IN A BIOLOGICAL SPECIMEN COMPRISING THE MEASUREMENT OF GLUTATHIONE-S-TRANSFERASE ENZYMATIC ACTIVITY IN THE PRESENCE AND ABSENCE AN AMOUNT OF A COMPOUND OF THE FORMULA HALO THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2002-12-17 US disclosed
US-6103665-A Inhibition of glutathione transferase by haloenol lactones THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-08-15 US disclosed
US-5767147-A MEDICAL DIAGNOSIS, TREATMENT OF DRUG RESISTANCE IN CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-06-16 US disclosed
WO-1996032936-A1 INHIBITION OF GLUTATHIONE TRANSFERASE BY HALOENOL LACTONES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-10-24 WO disclosed