SCHEMBL765607

SCHEMBL765607

CCC(C)c1ccccc1Oc1ccc(CN)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.43
SLC6A4 P31645 4/20 0.43
ST14 Q9Y5Y6 1/20 0.43
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 1/20 0.40
DPP4 P27487 1/20 0.40
NISCH Q9Y2I1 1/20 0.39
CARM1 Q86X55 2/20 0.39
PRMT6 Q96LA8 2/20 0.39
HTT P42858 2/20 0.39
MAOB P27338 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
KCNH2 Q12809 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506593 0.86 ST14 (0.47) HTR2ASLC6A4ST14L3MBTL1DPP4
SCHEMBL6680297 0.84 TSHR (0.50) HTR2ASLC6A4TSHRATML3MBTL1
SCHEMBL29960384 0.84 TSHR (0.50) HTR2ASLC6A4TSHRATML3MBTL1
SCHEMBL7710832 0.80 TSHR (0.57) HTR2ASLC6A4TSHRATML3MBTL1
SCHEMBL6061469 0.75 TSHR (0.49) HTR2ASLC6A4TSHRATML3MBTL1
SCHEMBL12239008 0.74 HRH1 (0.50) HTR2ASLC6A4ST14ATML3MBTL1
SCHEMBL5836321 0.74 HTR2A (0.61) HTR2ASLC6A4L3MBTL1KDM4EDPP4
SCHEMBL923365 0.74 HTT (0.70) SLC6A4ST14TSHRL3MBTL1DPP4
SCHEMBL507354 0.74 ST14 (0.52) ST14TSHRATML3MBTL1DPP4
SCHEMBL190108 0.73 TSHR (0.59) TSHRATML3MBTL1KDM4ENISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed