SCHEMBL765656

SCHEMBL765656

Bc1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4cncnc4)CC3)cc2)c(C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 5/20 0.49
MAPK14 Q16539 4/20 0.44
CYP3A4 P08684 1/20 0.44
UCHL1 P09936 1/20 0.35
VNN1 O95497 1/20 0.34
CTSL P07711 1/20 0.34
KDM1A O60341 1/20 0.34
HDAC1 Q13547 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
CTSK P43235 1/20 0.33
PTGER4 P35408 1/20 0.33
PTGER2 P43116 1/20 0.33
PLA2G7 Q13093 1/20 0.33
CNR1 P21554 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764428 0.90 BDKRB1 (0.51) BDKRB1MAPK14CYP3A4VNN1CTSL
SCHEMBL764449 0.90 BDKRB1 (0.49) BDKRB1MAPK14CYP3A4PTGDR2PTGER4
SCHEMBL764480 0.90 BDKRB1 (0.53) BDKRB1MAPK14CYP3A4VNN1KDM1A
SCHEMBL765805 0.90 BDKRB1 (0.49) BDKRB1MAPK14CYP3A4CTSLPTGDR2
SCHEMBL765846 0.90 BDKRB1 (0.49) BDKRB1MAPK14CYP3A4UCHL1VNN1
SCHEMBL765845 0.88 MAPK14 (0.58) BDKRB1MAPK14CYP3A4UCHL1CTSL
SCHEMBL765145 0.87 BDKRB1 (0.48) BDKRB1MAPK14CYP3A4KDM1AHDAC1
SCHEMBL13904099 0.87 BDKRB1 (0.51) BDKRB1MAPK14CYP3A4KDM1AHDAC1
SCHEMBL13904097 0.84 BDKRB1 (0.49) BDKRB1MAPK14CYP3A4KDM1AHDAC1
SCHEMBL765204 0.81 BDKRB1 (0.51) BDKRB1MAPK14CYP3A4PTGER4PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed