SCHEMBL7656622

SCHEMBL7656622

Nc1cccc2c1C(=O)CCC2N1C(=O)c2ccccc2C1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 12/20 0.59
DDB1 Q16531 11/20 0.59
IKZF3 Q9UKT9 3/20 0.59
TNF P01375 2/20 0.59
IL1B P01584 2/20 0.59
IKZF1 Q13422 2/20 0.59
TBXA2R P21731 1/20 0.59
ALDH1A1 P00352 1/20 0.48
CHRM2 P08172 1/20 0.48
OPRM1 P35372 1/20 0.48
CYP1A2 P05177 1/20 0.48
TSHR P16473 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TMEM97 Q5BJF2 3/20 0.43
HTR2B P41595 2/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1265364 0.81 CRBN (0.57) CRBNDDB1IKZF3TNFIL1B
SCHEMBL30998375 0.81 CRBN (0.57) CRBNDDB1IKZF3TNFIL1B
SCHEMBL1265365 0.81 CRBN (0.57) CRBNDDB1IKZF3TNFIL1B
SCHEMBL7650425 0.78 CRBN (0.50) CRBNDDB1IKZF3TNFIL1B
SCHEMBL7655805 0.77 DDB1 (0.49) CRBNDDB1IKZF3TNFIL1B
SCHEMBL7662576 0.77 DDB1 (0.49) CRBNDDB1IKZF3TNFIL1B
SCHEMBL7661705 0.76 DDB1 (0.63) CRBNDDB1IKZF3ALDH1A1CHRM2
SCHEMBL7664386 0.75 DDB1 (0.46) CRBNDDB1IKZF3TNFIL1B
SCHEMBL30703123 0.74 CRBN (0.57) CRBNDDB1IKZF3TNFIL1B
SCHEMBL2557698 0.74 CRBN (0.57) CRBNDDB1IKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407115-B1 ANTICARCINOGENIC AND ANTITUMOR AGENTS; SIDE EFFECT REDUCTION, WATER SOLUBILITY DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2002-06-18 US disclosed
US-5834476-A DERIVATIVE OF CAMPTOTHECIN, ANTITUMOR AGENT, ANTICARCINOGENIC AGENT DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-11-10 US disclosed
US-5770605-A Method for treating leukemia with a hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-06-23 US disclosed
US-5658920-A ANTITUMOR AGENTS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-08-19 US disclosed
US-5637770-A Hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-06-10 US disclosed
EP-0495432-B1 Hexa-cyclic compound DAIICHI SEIYAKU CO (JP) 1996-05-29 EP disclosed
EP-0495432-A1 Hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1992-07-22 EP disclosed