SCHEMBL7656904

SCHEMBL7656904

COc1ccc(C(=O)CC(=O)CC(=O)O)cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA4 P22748 1/20 0.59
CA6 P23280 1/20 0.59
CA7 P43166 1/20 0.59
TPMT P51580 1/20 0.59
CA9 Q16790 1/20 0.59
CA14 Q9ULX7 1/20 0.59
MAPT P10636 4/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
ALDH1A1 P00352 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
GAA P10253 1/20 0.57
TSHR P16473 3/20 0.56
CTNNB1 P35222 2/20 0.56
WNT3A P56704 2/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL8416081 0.95 CA12 (0.54) CA12CA1CA2CA4CA6
SCHEMBL30629388 0.92 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL4438295 0.92 CA12 (0.65) CA12CA1CA2CA4CA6
SCHEMBL7659731 0.87 MAPT (0.57) CA12CA1CA2CA4CA6
SCHEMBL1659363 0.86 MAPT (0.71) CA12CA1CA2CA4CA6
SCHEMBL29668496 0.82 MEN1 (0.71) CA12CA1CA2CA4CA6
SCHEMBL28881824 0.82 MEN1 (0.71) CA12CA1CA2CA4CA6
SCHEMBL11045656 0.81 MAPT (0.61) CA12CA1CA2CA4CA6
SCHEMBL1322947 0.81 MAPT (0.61) CA12CA1CA2CA4CA6
SCHEMBL7380780 0.81 MAPT (0.61) CA12CA1CA2CA4CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6384045-B1 TREATMENT OF ALZHEIMER'S DISEASE AND ANTICANCER AGENTS KANSAS STATE UNIVERSITY RESEARCH FOUNDATION 2002-05-07 US disclosed
US-5958970-A ENZYME INHIBITORS OF ACETYLCHOLINESTERASE (ACHE) AND ACYL-COA:CHOLESTEROL ACYLTRANSFERASE (ACAT); USED IN THE TREATMENT OF ALZHEIMER'S DISEASE, ATHEROSCLEROSIS AND HYPERCHOLESTEROLEMIA KANSAS STATE UNIVERSITY RESEARCH FOUNDATION (US) 1999-09-28 US disclosed
WO-1998039010-A1 TRICYCLIC AND TETRACYCLIC PYRONES KANSAS STATE UNIVERSITY RESEARCH FOUNDATION (US) 1998-09-11 WO disclosed