SCHEMBL7657253

SCHEMBL7657253

CCCCc1c[nH]c(Cc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.40
TAAR1 Q96RJ0 1/20 0.40
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
PARP1 P09874 1/20 0.39
KCNH2 Q12809 1/20 0.39
TLR7 Q9NYK1 3/20 0.38
GAA P10253 1/20 0.38
HSD11B1 P28845 1/20 0.38
CYP19A1 P11511 3/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15147961 0.95 KCNH2 (0.45) TLR8TAAR1KCNH2HSD11B1CYP19A1
SCHEMBL28016575 0.94 KCNH2 (0.47) TLR8KCNH2TLR7CYP19A1NPC1
Ammonia Solution, Strong SCHEMBL27918102 0.93 KCNH2 (0.46) TLR8KCNH2TLR7CYP19A1NPC1
SCHEMBL7665114 0.90 TAAR1 (0.42) TAAR1ADORA2AGAACYP19A1NR1H2
SCHEMBL27864776 0.89 CYP19A1 (0.44) TLR8KCNH2TLR7CYP19A1NPC1
SCHEMBL9214238 0.88 TLR8 (0.43) TLR8TAAR1ADORA3ADORA2APARP1
Ethylene SCHEMBL28202240 0.84 TLR8 (0.43) TLR8TAAR1ADORA3ADORA2APARP1
SCHEMBL28356909 0.83 KCNH2 (0.50) TAAR1KCNH2GAANR1H2NR1H3
Biphenyl SCHEMBL7417032 0.83 PARP1 (0.43) ADORA3ADORA2APARP1KCNH2HSD11B1
SCHEMBL1723556 0.81 TAAR1 (0.48) TAAR1ADORA2AGAANR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492377-B1 Imidazotriazolopyrimidines with adenosine-antagonistic activity BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-10 US disclosed