SCHEMBL7657372

SCHEMBL7657372

COC(=O)Cn1c(=O)c2ccccc2n(CCCCCl)c1=O

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.57
KDM4E B2RXH2 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
KMT2A Q03164 2/20 0.49
TP53 P04637 1/20 0.48
TNF P01375 1/20 0.46
S1PR2 O95136 1/20 0.46
MAPT P10636 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPK1 P28482 1/20 0.46
MDM2 Q00987 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649581 0.96 CNR2 (0.56) CNR2KDM4ESMN1; SMN2KMT2ATP53
SCHEMBL7650022 0.81 TNF (0.73) CNR2TP53TNF
SCHEMBL7656518 0.81 TNF (0.67) CNR2KDM4ETP53TNF
SCHEMBL7649598 0.78 TSHR (0.55) CNR2KDM4ESMN1; SMN2KMT2ATNF
SCHEMBL7653389 0.78 P2RX4 (0.60) SMN1; SMN2KMT2ATP53MAPT
SCHEMBL25936310 0.77 KDM4E (0.61) CNR2KDM4ESMN1; SMN2KMT2ATP53
SCHEMBL7650027 0.77 TNF (0.68) CNR2KDM4EKMT2ATNF
SCHEMBL7652923 0.77 P2RX4 (0.58) SMN1; SMN2KMT2ATP53MAPT
SCHEMBL7652144 0.76 BCHE (0.51) CNR2KMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL5037066 0.75 TNF (0.59) CNR2KDM4ESMN1; SMN2KMT2ATNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed