SCHEMBL765822

SCHEMBL765822

O=C(NC1(C(=O)NCc2ccc(Oc3cc(C(F)F)cc(C(F)(F)F)c3)cc2)CC1)c1cncnc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 5/20 0.49
MAPK14 Q16539 3/20 0.41
USP36 Q9P275 1/20 0.40
CCR2 P41597 2/20 0.36
KCNH2 Q12809 2/20 0.36
S1PR2 O95136 1/20 0.36
CNR1 P21554 1/20 0.36
KDM1A O60341 1/20 0.35
HDAC1 Q13547 1/20 0.35
SCN9A Q15858 1/20 0.35
CXCR4 P61073 1/20 0.35
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764448 0.92 BDKRB1 (0.53) BDKRB1MAPK14USP36CCR2KCNH2
SCHEMBL12239075 0.88 BDKRB1 (0.52) BDKRB1MAPK14USP36CCR2KCNH2
SCHEMBL765169 0.87 BDKRB1 (0.55) BDKRB1MAPK14KDM1AHDAC1CYP3A4
SCHEMBL10121171 0.84 BDKRB1 (0.46) BDKRB1MAPK14USP36CCR2KCNH2
SCHEMBL12239076 0.82 BDKRB1 (0.56) BDKRB1MAPK14CYP3A4
SCHEMBL12262778 0.82 BDKRB1 (0.58) BDKRB1MAPK14HDAC1
SCHEMBL10121362 0.81 BDKRB1 (0.58) BDKRB1MAPK14SCN9ACXCR4CYP3A4
SCHEMBL13904174 0.80 BDKRB1 (0.49) BDKRB1MAPK14USP36CCR2KCNH2
SCHEMBL765145 0.80 BDKRB1 (0.48) BDKRB1MAPK14KDM1AHDAC1SCN9A
SCHEMBL764413 0.80 BDKRB1 (0.64) BDKRB1MAPK14CNR1HDAC1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed